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Drug

Chenodeoxycholic Acid

Approved · EMA
ClassBile acid receptor FXR agonistEmerging researchLate-stage development
Also known as 3alpha,7alpha-Dihydroxy-5beta-cholanic acid, Acide chenodeoxycholique, Acido chenodeoxicholico, Acidum chenodeoxycholicum+10 more

3alpha,7alpha-Dihydroxy-5beta-cholanic acid, Acide chenodeoxycholique, Acido chenodeoxicholico, Acidum chenodeoxycholicum, Anthropodeoxycholic acid, Anthropodesoxycholic acid, CDCA, CDCA - chenodeoxycholic acid, CHENODIOL, Chenic acid, Chenocholic acid, Gallodesoxycholic acid, Chenodesoxycholic acid, 3 alpha,7 alpha, dihydroxycholanic acid.

2
Research papers
Bile acid receptor
Primary target
1
Regulatory events
Latest activity
beta

Recent clinical, regulatory, research and industry developments relating to this drug.

Changes in Bile Acid Homeostasis and Stool Habits After Cholecystectomy

Clinical trial2022-05-19Results posted · ClinicalTrials.gov

Biologic Significance of Cholestanol in Man

Clinical trial2009-12-01Withdrawn · ClinicalTrials.gov

Profile

Identifiers & mechanism

Canonical identifiers, marketed brand names and mechanism, resolved across RxNorm, ChEMBL and ATC.

Canonical name
Chenodeoxycholic Acid
Aliases & brands
3alpha,7alpha-Dihydroxy-5beta-cholanic acidAcide chenodeoxycholiqueAcido chenodeoxicholicoAcidum chenodeoxycholicumAnthropodeoxycholic acidAnthropodesoxycholic acidCDCACDCA - chenodeoxycholic acidCHENODIOLChenic acidChenocholic acidGallodesoxycholic acidChenodesoxycholic acid3 alpha,7 alpha, dihydroxycholanic acid
RxNorm CUI
2323
ChEMBL ID
CHEMBL240597
ATC codes
A05AA01
UNII
0GEI24LG0J
Primary mechanism
Bile acid receptor FXR agonist
Regulatory jurisdictions
ema

Pharmacology & targets

1 target

Known molecular targets and mechanisms supported by curated pharmacology databases.

Bile acid receptor
NR1H4 · Q96RI1
AGONISTBile acid receptor FXR agonist

Regulatory timeline

1 event

The complete regulatory record, grouped by authority — approvals, safety advisories and label changes. Each authority shows its most recent events; expand one to read its full history.

Earliest approval
2017-04-10
Latest approval
2017-04-10
Authorities
EMA
Total events
1
emaEuropean Medicines Agency· 1 event
2017-04-10Approval
Approval: Chenodeoxycholic acid Leadiant (previously Chenodeoxycholic acid sigma-tau) (EMA)
Indication: Chenodeoxycholic acid is indicated for the treatment of inborn errors of primary bile acid synthesis due to sterol 27 hydroxylase deficiency (presenting as cerebrotendinousShow full indication

Chenodeoxycholic acid is indicated for the treatment of inborn errors of primary bile acid synthesis due to sterol 27 hydroxylase deficiency (presenting as cerebrotendinous xanthomatosis (CTX)) in infants, children and adolescents aged 1 month to 18 years and adults.

Evidence ↗

Contains information from the European Medicines Agency (European Medicines Agency), © EMA, reused under CC BY 4.0.

Clinical trials

11 trials

The current development programme across all trial phases — status mix, phase distribution and the late-stage studies shaping the evidence base.

Development programme
CLINICALTRIALS.GOV · LIVE REGISTRY
11
registered trials across all phases
LATEST COMPLETION 2022
8
Late-stage (III+)
7
Completed
4
Discontinued
PHASE DISTRIBUTIONn = 11
Early Phase 11Phase 11Phase 21Phase 31Phase 44Phase N / A3

Late-stage studies

Phase III+ trials still open or recently active — where late-stage evidence is being generated.

Recent completions

Trials that read out recently, adding to the completed evidence base.

Research activity

2 papers

Key research shaping understanding of this drug, combining the latest publications with the most influential evidence.

Publications over time
20192020
Major research themes3
Fermented Foods1Gastrointestinal Microbiome1Tea1
Journals, researchers & institutions
Top journals
  • EBioMedicine1
  • Nature communications1
Leading researchers
  • Bian Z2
  • Han X2
  • Huang F2
  • Jia W2
  • Li M2
  • Rajani C2
  • Wang S2
  • Wei M2
Leading institutions
free-text, unnormalised
  • Chinese Medicine Clinical Study Center1
  • Functional Metabolomic and Gut Microbiome Laboratory1
  • School of Chinese Medicine1
  • School of Pharmacy1
  • Shanghai Jiao Tong University Affiliated Six People's Hospital1
  • Shanghai Key Laboratory of Diabetes Mellitus and Center for Translational Medicine1

Related drugs

3 matches

Drugs sharing diseases, protein targets and literature with this one. Ranked by graph evidence (shared targets + diseases weighted above co-mentions).

Acts on the same molecular target as Chenodeoxycholic Acid, with 3 overlapping disease areas.

Shared target3 shared diseases1 shared paper

Studied across 3 of the same disease areas as Chenodeoxycholic Acid in the shared literature.

3 shared diseases1 shared paper

Studied across 2 of the same disease areas as Chenodeoxycholic Acid in the shared literature.

2 shared diseases1 shared paper
References & data sources
  • RxNorm (U.S. National Library of Medicine) — drug identity
  • ChEMBL (EMBL-EBI) & UniProt — pharmacology and targets
  • Europe PMC — research literature
  • ClinicalTrials.gov — clinical trials
  • Regulatory event sources are credited in the Regulatory Timeline above.