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Drug

Amivantamab

Approved · EMA
ClassEpidermal growth factor receptor erbB1 inhibitorEmerging researchLate-stage development

Also known as Rybrevant, Rybrevant Faspro.

2
Research papers
33
Active clinical trials
2
Protein targets
1
Regulatory events
Latest activity
beta

Recent clinical, regulatory, research and industry developments relating to this drug.

Approval: Rybrevant (EMA)

Regulatory2021-12-09EMA

Amivantamab in EGFR Exon 20 Insertion-Mutated Non-Small-Cell Lung Cancer Progressing on Platinum Chemotherapy: Initial Results From the CHRYSALIS Phase I Study.

Research2021-08-02Journal of clinical oncology : official journal of the American Society of Clinical Oncology

Profile

Identifiers & mechanism

Canonical identifiers, marketed brand names and mechanism, resolved across RxNorm, ChEMBL and ATC.

Canonical name
Amivantamab
Aliases & brands
RybrevantRybrevant Faspro
RxNorm CUI
2549199
ChEMBL ID
CHEMBL4297774
ATC codes
L01FX18
UNII
0JSR7Z0NB6
Primary mechanism
Epidermal growth factor receptor erbB1 inhibitor
Regulatory jurisdictions
ema

Pharmacology & targets

2 targets

Known molecular targets and mechanisms supported by curated pharmacology databases.

INHIBITOREpidermal growth factor receptor erbB1 inhibitor
INHIBITORHepatocyte growth factor receptor inhibitor

Regulatory timeline

1 event

The complete regulatory record, grouped by authority — approvals, safety advisories and label changes. Each authority shows its most recent events; expand one to read its full history.

Earliest approval
2021-12-09
Latest approval
2021-12-09
Authorities
EMA
Total events
1
emaEuropean Medicines Agency· 1 event
2021-12-09Approval
Approval: Rybrevant (EMA)
Indication: Rybrevant is indicated: in combination with lazertinib for the first line treatment of adult patients with advanced non small cell lung cancer (NSCLC) with EGFR Exon 19 deletionsShow full indication

Rybrevant is indicated: in combination with lazertinib for the first line treatment of adult patients with advanced non small cell lung cancer (NSCLC) with EGFR Exon 19 deletions or Exon 21 L858R substitution mutations. in combination with carboplatin and pemetrexed for the treatment of adult patients with advanced NSCLC with EGFR Exon 19 deletions or Exon 21 L858R substitution mutations after failure of prior therapy including an EGFR tyrosine kinase inhibitor (TKI). in combination with carboplatin and pemetrexed for the first line treatment of adult patients with advanced NSCLC with activating EGFR Exon 20 insertion mutations. as monotherapy for treatment of adult patients with advanced NSCLC with activating EGFR Exon 20 insertion mutations, after failure of platinum based therapy.

Evidence ↗

Contains information from the European Medicines Agency (European Medicines Agency), © EMA, reused under CC BY 4.0.

Clinical trials

38 trials

The current development programme across all trial phases — status mix, phase distribution and the late-stage studies shaping the evidence base.

Development programme
CLINICALTRIALS.GOV · LIVE REGISTRY
38
registered trials across all phases
LATEST COMPLETION 2026
33
Active studies
16
Recruiting
7
Late-stage (III+)
2
Completed
3
Discontinued
PHASE DISTRIBUTIONn = 38
Phase 15Phase 1 / 28Phase 218Phase 37

Late-stage studies

Phase III+ trials still open or recently active — where late-stage evidence is being generated.

Recent completions

Trials that read out recently, adding to the completed evidence base.

Research activity

2 papers

Key research shaping understanding of this drug, combining the latest publications with the most influential evidence.

Publications over time
20212024
Most influential

Amivantamab in EGFR Exon 20 Insertion-Mutated Non-Small-Cell Lung Cancer Progressing on Platinum Chemotherapy: Initial Results From the CHRYSALIS Phase I Study.

Journal of clinical oncology : official journal of the American Society of Clinical Oncology · 2021 · 499 cites
Recent papers

Amivantamab in EGFR Exon 20 Insertion-Mutated Non-Small-Cell Lung Cancer Progressing on Platinum Chemotherapy: Initial Results From the CHRYSALIS Phase I Study.

Journal of clinical oncology : official journal of the American Society of Clinical Oncology · 2021 · 499 cites
Major research themes7
Antibodies, Bispecific1Antineoplastic Combined Chemotherapy Protocols1Carcinoma, Non-Small-Cell Lung1Lung Neoplasms1Morpholines1Pyrazoles1Pyrimidines1
Journals, researchers & institutions
Top journals
  • Journal of clinical oncology : official journal of the American Society of Clinical Oncology1
  • The New England journal of medicine1
Leading researchers
  • Bauml JM2
  • Cho BC2
  • Girard N2
  • Kim SW2
  • Knoblauch RE2
  • Lee JS2
  • Lee KH2
  • Lorenzini P2
Leading institutions
free-text, unnormalised
  • Yonsei Cancer Center2
  • Asan Medical Center1
  • Chungbuk National University Hospital1
  • City of Hope Comprehensive Cancer Center1
  • Columbia University Medical Center1
  • Earle A. Chiles Research Institute1

Related diseases

2 conditions

Regulator-approved indications and conditions co-mentioned with this drug across the research literature. Number shows shared papers.

Related drugs

2 matches

Drugs sharing diseases, protein targets and literature with this one. Ranked by graph evidence (shared targets + diseases weighted above co-mentions).

Acts on the same molecular target as Amivantamab, with 2 overlapping disease areas.

Shared target2 shared diseases1 shared paper

Acts on the same molecular target as Amivantamab, with 2 overlapping disease areas.

Shared target2 shared diseases1 shared paper
References & data sources
  • RxNorm (U.S. National Library of Medicine) — drug identity
  • ChEMBL (EMBL-EBI) & UniProt — pharmacology and targets
  • Europe PMC — research literature
  • ClinicalTrials.gov — clinical trials
  • Regulatory event sources are credited in the Regulatory Timeline above.