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Drug

Tezacaftor

In clinical development
ClassCystic fibrosis transmembrane conductance regulator positive modulatorEmerging researchEarly-to-mid development

Also known as Alyftrek.

1
Research papers
1
Active clinical trials
CFTR
Primary target
Latest activity
beta

Recent clinical, regulatory, research and industry developments relating to this drug.

Profile

Identifiers & mechanism

Canonical identifiers, marketed brand names and mechanism, resolved across RxNorm, ChEMBL and ATC.

Canonical name
Tezacaftor
Aliases & brands
Alyftrek
RxNorm CUI
1999382
ChEMBL ID
CHEMBL3544914
UNII
8RW88Y506K
Primary mechanism
Cystic fibrosis transmembrane conductance regulator positive modulator

Pharmacology & targets

1 target

Known molecular targets and mechanisms supported by curated pharmacology databases.

POSITIVE MODULATORCystic fibrosis transmembrane conductance regulator positive modulator

Clinical trials

2 trials

The current development programme across all trial phases — status mix, phase distribution and the late-stage studies shaping the evidence base.

Development programme
CLINICALTRIALS.GOV · LIVE REGISTRY
2
registered trials across all phases
LATEST COMPLETION 2017
1
Active studies
1
Completed
PHASE DISTRIBUTIONn = 2
Phase 12

Recent completions

Trials that read out recently, adding to the completed evidence base.

Research activity

1 papers

Key research shaping understanding of this drug, combining the latest publications with the most influential evidence.

Major research themes1
Cystic Fibrosis1
Journals, researchers & institutions
Top journals
  • Respiratory research1
Leading researchers
  • Conrad D1
  • Gil M1
  • Gonzalez CT1
  • Guzior DV1
  • Martin C1
  • McClelland M1
  • Mielke J1
  • Okros M1
Leading institutions
free-text, unnormalised
  • Medical University of Vienna1
  • Michigan State University1
  • University of California San Diego1

Related drugs

2 matches

Drugs sharing diseases, protein targets and literature with this one. Ranked by graph evidence (shared targets + diseases weighted above co-mentions).

Acts on the same molecular target as Tezacaftor, with an overlapping disease area.

Shared target1 shared disease1 shared paper

Acts on the same molecular target as Tezacaftor, with an overlapping disease area.

Shared target1 shared disease1 shared paper
References & data sources
  • RxNorm (U.S. National Library of Medicine) — drug identity
  • ChEMBL (EMBL-EBI) & UniProt — pharmacology and targets
  • Europe PMC — research literature
  • ClinicalTrials.gov — clinical trials